Small Molecule Modulators of β-arrestins.

Kahsai AW, Pakharukova N, Kwon HY, Shah KS, del Real CT, Shreiber BN, Liang-Lin JG, Shim PJ, Lee MA, Ngo VA, Schwalb AM, Pham U, Chundi A, Jiang H, Flores-Espinoza E, Liu S, Nibley PC, Bassford DK, Hahn H, Kunzle CA, Thomas BN, Kim J, Zhou Y, Wang J, Zhang X, Smith JS, Rein LAM, Thomsen ARB, Shenoy SK, Rajagopal S, Shi L, Ahn S, Rockman HA, Masoudi A, Lefkowitz RJ (2026). Nature 656, 770–779.

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Alex Thomsen
Distinct Conformations of GPCR–β-Arrestin Complexes Mediate Desensitization, Signaling and Endocytosis

Cahill III TJ*, Thomsen ARB*, Tarrasch JT, Plouffe B, Nguyen A, Yang F, Bassoni D, Gavino B, Lamerdin J, Triest S, Huang L-Y, Shukla A, Kahsai AW, Berger B, Little IV J, Antar A, Blanc A, Qu C-X, Chen X, Kawakami K, Inoue A, Aoki J, Steyeart J, Sun J-P, Bouvier M, Skiniotis G, Lefkowitz RJ (2017). Proceedings of the National Academy of Sciences USA, 114:2562-67.
*co-first authors

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